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1 . Academic Journal
Identification by High-Throughput Screening of Pseudomonas Acyl–Coenzyme A Synthetase Inhibitors
저자
by
Turcano, Lorenzo
;
Visaggio, Daniela
;
Frangipani, Emanuela
;
Missineo, Antonino
;
Andreini, Matteo
, et al.
소스
In
SLAS Discovery
August 2017 22(7):897-905
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7 . Academic Journal
Structure–activity relationship and properties optimization of a series of Quinazoline-2,4-diones as inhibitors of the canonical Wnt pathway
저자
by
Nencini, Arianna
;
Pratelli, Carmela
;
Quinn, Joanna M.
;
Salerno, Massimiliano
;
Tunici, Patrizia
, et al.
소스
In
European Journal of Medicinal Chemistry
5 May 2015 95:526-545
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7 . Academic Journal
Peptidomimetic nitrile inhibitors of malarial protease falcipain-2 with high selectivity against human cathepsins
저자
by
Nizi, Emanuela
;
Sferrazza, Alessio
;
Fabbrini, Danilo
;
Nardi, Valentina
;
Andreini, Matteo
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 May 2018 28(9):1540-1544
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7 . Academic Journal
BACE1 inhibitors: A head group scan on a series of amides
저자
by
Woltering, Thomas J.
;
Wostl, Wolfgang
;
Hilpert, Hans
;
Rogers-Evans, Mark
;
Pinard, Emmanuel
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 July 2013 23(14):4239-4243
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7 . Academic Journal
Identification and binding mode of a novel Leishmania Trypanothione reductase inhibitor from high throughput screening.
저자
by
Turcano, Lorenzo
;
Torrente, Esther
;
Missineo, Antonino
;
Andreini, Matteo
;
Gramiccia, Marina
, et al.
소스
PLoS Neglected Tropical Diseases
. 11/26/2018, Vol. 12 Issue 11, p1-21. 21p.
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7 . Academic Journal
Discovery by organism based high-throughput screening of new multi-stage compounds affecting Schistosoma mansoni viability, egg formation and production.
저자
by
Guidi, Alessandra
;
Lalli, Cristiana
;
Gimmelli, Roberto
;
Nizi, Emanuela
;
Andreini, Matteo
, et al.
소스
PLoS Neglected Tropical Diseases
. 10/6/2017, Vol. 11 Issue 10, p1-21. 21p.
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7 . Academic Journal
Optimization of linear and cyclic peptide inhibitors of KEAP1-NRF2 protein-protein interaction
저자
by
Colarusso, Stefania
;
De Simone, Daniele
;
Frattarelli, Tommaso
;
Andreini, Matteo
;
Cerretani, Mauro
, et al.
소스
BIOORGANIC & MEDICINAL CHEMISTRY
; NOV 1 2020, 28 21, p115738 12p.
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7 . Academic Journal
Combined Peptide and Small-Molecule Approach toward Nonacidic THIQ Inhibitors of the KEAP1/NRF2 Interaction
저자
by
Ontoria, Jesus M.
;
Biancofiore, Ilaria
;
Fezzardi, Paola
;
Ferrigno, Federica
;
Torrente, Esther
, et al.
소스
ACS MEDICINAL CHEMISTRY LETTERS
; MAY 14 2020, 11 5, p740-p746, 7p.
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7 . Periodical
Identification by High-Throughput Screening of PseudomonasAcyl–Coenzyme A Synthetase Inhibitors
저자
by
Turcano, Lorenzo
;
Visaggio, Daniela
;
Frangipani, Emanuela
;
Missineo, Antonino
;
Andreini, Matteo
, et al.
소스
Journal of Biomolecular Screening; August 2017, Vol. 22 Issue: 7 p897-905, 9p
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7 . Academic Journal
The soluble Y115E-Y117E variant of human glutaminyl cyclase is a valid target for X-ray and NMR screening of inhibitors against Alzheimer disease.
저자
by
DiPisa, Flavio
;
Pozzi, Cecilia
;
Benvenuti, Manuela
;
Andreini, Matteo
;
Marconi, Guido
, et al.
소스
Acta Crystallographica: Section F, Structural Biology Communications
. Aug2015, Vol. 71 Issue 8, p986-992. 7p.
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