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1 . Academic Journal
Small molecule branched-chain ketoacid dehydrogenase kinase (BDK) inhibitors with opposing effects on BDK protein levels
저자
by
Rachel J. Roth Flach
;
Eliza Bollinger
;
Allan R. Reyes
;
Brigitte Laforest
;
Bethany L. Kormos
, et al.
소스
Nature Communications, Vol 14, Iss 1, Pp 1-14 (2023)
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7 . Academic Journal
Crystal structure of human lysosomal acid lipase and its implications in cholesteryl ester storage disease[S]
저자
by
Francis Rajamohan
;
Allan R. Reyes
;
Meihua Tu
;
Nicole L. Nedoma
;
Lise R. Hoth
, et al.
소스
Journal of Lipid Research, Vol 61, Iss 8, Pp 1192-1202 (2020)
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7 .
Structural studies identify angiotensin II receptor blocker-like compounds as branched-chain ketoacid dehydrogenase kinase inhibitors
저자
by
Shenping Liu
;
Bethany L. Kormos
;
John D. Knafels
;
Parag V. Sahasrabudhe
;
Amy Rosado
, et al.
소스
Journal of Biological Chemistry
. 299:102959
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7 .
Crystal structure of human lysosomal acid lipase and its implications in cholesteryl ester storage disease[S]
저자
by
Adam G. Schwaid
;
Jessica Ward
;
Nicole L. Nedoma
;
Lise R. Hoth
;
Meihua Tu
, et al.
소스
Journal of Lipid Research, Vol 61, Iss 8, Pp 1192-1202 (2020)
Journal of Lipid Research
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7 .
Acyl Glucuronide Metabolites of 6-Chloro-5-[4-(1-hydroxycyclobutyl)phenyl]-1H-indole-3-carboxylic Acid (PF-06409577) and Related Indole-3-carboxylic Acid Derivatives are Direct Activators of Adenosine Monophosphate-Activated Protein Kinase (AMPK)
저자
by
Gregory S. Walker
;
Kimberly O. Cameron
;
Janice A. Brown
;
Daniel W. Kung
;
Angela Wolford
, et al.
소스
Journal of Medicinal Chemistry
. 61:7273-7288
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7 .
Activation of Liver AMPK with PF-06409577 Corrects NAFLD and Lowers Cholesterol in Rodent and Primate Preclinical Models
저자
by
Jessica Ward
;
Jason Barricklow
;
Chuong Nguyen
;
Eliza Bollinger
;
Christopher T. Salatto
, et al.
소스
EBioMedicine, Vol 31, Iss, Pp 122-132 (2018)
EBioMedicine
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7 .
Selective Activation of AMPKβ1-Containing Isoforms Improves Kidney Function in a Rat Model of Diabetic Nephropathy
저자
by
Paul DaSilva-Jardine
;
Jessica Ward
;
Katherine Cialdea
;
Matthew F. Calabrese
;
Marina Amaro
, et al.
소스
Journal of Pharmacology and Experimental Therapeutics
. 361:303-311
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7 .
Discovery and Preclinical Characterization of 6-Chloro-5-[4-(1-hydroxycyclobutyl)phenyl]-1H-indole-3-carboxylic Acid (PF-06409577), a Direct Activator of Adenosine Monophosphate-activated Protein Kinase (AMPK), for the Potential Treatment of Diabetic Nephropathy
저자
by
Jane M. Withka
;
Daniel W. Kung
;
Russell A. Miller
;
Matthew S. Dowling
;
Aaron C. Smith
, et al.
소스
Journal of Medicinal Chemistry
. 59:8068-8081
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7 .
Optimization of Metabolic and Renal Clearance in a Series of Indole Acid Direct Activators of 5'-Adenosine Monophosphate-Activated Protein Kinase (AMPK)
저자
by
Kimberly O. Cameron
;
Kevin J. Filipski
;
Jana Polivkova
;
Matthew S. Dowling
;
Andre Shavnya
, et al.
소스
Journal of medicinal chemistry
. 61(6)
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7 .
Biophysical Interactions of Direct AMPK Activators
저자
by
Jane M. Withka
;
Graham M. West
;
Kris A. Borzilleri
;
Ravi G. Kurumbail
;
Francis Rajamohan
, et al.
소스
Methods in Molecular Biology ISBN: 9781493975976
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