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1 .
Discovery and Optimization of 5-Amino-1,2,3-triazole-4-carboxamide Series against Trypanosoma cruzi
저자
by
Laste Stojanovski
;
Tania Bakshi
;
Iain H. Reid
;
Maria L. Marco
;
Stephen Brand
, et al.
소스
Journal of Medicinal Chemistry
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7 .
Use of Calculated Physicochemical Properties to Enhance Quantitative Response When Using Charged Aerosol Detection
저자
by
Richard J. Upton
;
Max W. Robinson
;
John C. Hollerton
;
Bob Boughtflower
;
Sean M. Lynn
, et al.
소스
Analytical Chemistry
. 89:1772-1777
Open Access (OpenAIRE)
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7 .
Synthesis and Structure–Activity Relationships of Indazole Arylsulfonamides as Allosteric CC-Chemokine Receptor 4 (CCR4) Antagonists
저자
by
Rebecca H. Graves
;
Alan P. Hill
;
David E. Clapham
;
Steven L. Sollis
;
Karen M. L. Morriss
, et al.
소스
Journal of Medicinal Chemistry
. 56:1946-1960
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7 .
Getting physical in drug discovery II: the impact of chromatographic hydrophobicity measurements and aromaticity
저자
by
Darren V. S. Green
;
Robert J. Young
;
Christopher N. Luscombe
;
Alan P. Hill
.
소스
Drug Discovery Today
. 16:822-830
Web of Science
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6 .
Estimating unbound volume of distribution and tissue binding by in vitro HPLC-based human serum albumin and immobilised artificial membrane-binding measurements
저자
by
Klára Valkó
;
Alan P. Hill
;
Shenaz Nunhuck
.
소스
Journal of pharmaceutical sciences
. 100(3)
Full Text (ScienceDirect)
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5 .
Getting physical in drug discovery: a contemporary perspective on solubility and hydrophobicity
저자
by
Alan P. Hill
;
Robert J. Young
.
소스
Drug discovery today
. 15(15-16)
Full Text (ScienceDirect)
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4 .
Dimeric zanamivir conjugates with various linking groups are potent, long-lasting inhibitors of influenza neuraminidase including H5N1 avian influenza
저자
by
Simon J. F. Macdonald
;
Alan P. Hill
;
Rob J. Fenton
;
Gail Mills
;
Stephanie Hamilton
, et al.
소스
Journal of medicinal chemistry
. 48(8)
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7 .
pKa prediction in multiply-substituted phenols: A comparison of multiple linear regression and back-propagation
저자
by
Valerie S. Rose
;
Richard Martin Hyde
;
Anne Hersey
;
Alan P. Hill
.
소스
Trends in QSAR and Molecular Modelling 92 ISBN: 9789072199133
Trends in QSAR and Molecular Modelling 92
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6 .
Principles of Method Selection in Partition Studies
저자
by
Alan P. Hill
;
David J. Livingstone
;
Richard Martin Hyde
;
Anne Hersey
.
소스
Quantitative Structure-Activity Relationships
. 8:288-296
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