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1 .
ACAT-selective and Nonselective DGAT1 Inhibition
저자
by
Tim J.D. Smith
;
Alan Martin Birch
;
Andrew V. Turnbull
;
Huw B. Jones
;
Linda K. Buckett
, et al.
소스
Toxicologic Pathology
. 41:941-950
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7 .
Discovery and optimization of efficacious neutral 4-amino-6-biphenyl-7,8-dihydropyrimido[5,4-f][1,4]oxazepin-5-one diacylglycerol acyl transferase-1 (DGAT1) inhibitors
저자
by
Frederick W. Goldberg
;
Alan Martin Birch
;
Andrew G. Leach
;
Wendy L. Snelson
;
Linda K. Buckett
, et al.
소스
MedChemComm
. 4:165-174
Scopus
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7 .
Optimisation of aqueous solubility in a series of G protein coupled receptor 119 (GPR119) agonists
저자
by
Katy J. Brocklehurst
;
Paul Schofield
;
James S. Scott
;
Per H. Svensson
;
Sam D. Groombridge
, et al.
소스
MedChemComm
. 4:95-100
Scopus
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7 .
Use of Small-Molecule Crystal Structures To Address Solubility in a Novel Series of G Protein Coupled Receptor 119 Agonists: Optimization of a Lead and in Vivo Evaluation
저자
by
David S. Clarke
;
Adrian Pickup
;
Andrew G. Leach
;
Pernilla Sörme
;
James S. Scott
, et al.
소스
Journal of Medicinal Chemistry
. 55:5361-5379
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7 .
Rationally Designing Safer Anilines: The Challenging Case of 4-Aminobiphenyls
저자
by
Robert P. Law
;
Carolin Schramm
;
Christine Mee
;
Andrew G. Leach
;
Sam D. Groombridge
, et al.
소스
Journal of Medicinal Chemistry
. 55:3923-3933
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7 .
Expedient Syntheses of Sulfonylhydantoins and Two Six-Membered Analogues
저자
by
Alan Martin Birch
;
Andrew D. Campell
.
소스
Synlett
. :0834-0838
Web of Science
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4 .
Identification, optimisation and in vivo evaluation of oxadiazole DGAT-1 inhibitors for the treatment of obesity and diabetes
저자
by
Graeme C. Moody
;
Alleyn T. Plowright
;
J. Matthew Wood
;
Matthew S. Addie
;
Scott Boyd
, et al.
소스
Bioorganicmedicinal chemistry letters
. 22(12)
Full Text (ScienceDirect)
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7 .
Discovery of a potent, selective, and orally efficacious pyrimidinooxazinyl bicyclooctaneacetic acid diacylglycerol acyltransferase-1 inhibitor
저자
by
Steven Wang
;
Susan Birtles
;
Graham J. Smith
;
Linda K. Buckett
;
Paul D. Kemmitt
, et al.
소스
Journal of medicinal chemistry
. 52(6)
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7 .
Matched molecular pair analysis of activity and properties of glycogen phosphorylase inhibitors
저자
by
Peter W. Kenny
;
Iain Simpson
;
Paul Robert Owen Whittamore
;
Alan Martin Birch
.
소스
Bioorganicmedicinal chemistry letters
. 19(3)
Full Text (ScienceDirect)
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6 .
Development of potent, orally active 1-substituted-3,4-dihydro-2-quinolone glycogen phosphorylase inhibitors
저자
by
Paul Robert Owen Whittamore
;
Nikos G. Oikonomakos
;
Peter W. Kenny
;
Dave P. Whalley
;
Ludovic Otterbein
, et al.
소스
Bioorganicmedicinal chemistry letters
. 17(2)
Full Text (ScienceDirect)
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