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1 . Academic Journal
Synthesis and biological evaluation of tert-butyl ester and ethyl ester prodrugs of L-γ-methyleneglutamic acid amides for cancer
저자
by
Khan, Md Imdadul H.
;
Mahdi, Fakhri
;
Penfornis, Patrice
;
Akins, Nicholas S.
;
Hossain, Md Imran
, et al.
소스
In
Bioorganic & Medicinal Chemistry
15 January 2023 78
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7 . Academic Journal
A systematic review on the kappa opioid receptor and its ligands: New directions for the treatment of pain, anxiety, depression, and drug abuse
저자
by
Khan, Md Imdadul H.
;
Sawyer, Benjamin J.
;
Akins, Nicholas S.
;
Le, Hoang V.
.
소스
In
European Journal of Medicinal Chemistry
5 December 2022 243
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6 . Academic Journal
Molecular mechanism of ligand gating and opening of NMDA receptor.
저자
by
Chou, Tsung-Han
;
Epstein, Max
;
Fritzemeier, Russell G.
;
Akins, Nicholas S.
;
Paladugu, Srinu
, et al.
소스
Nature; Aug2024, Vol. 632 Issue 8023, p209-217, 9p
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7 . Academic Journal
Development of a Dihydroquinoline–Pyrazoline GluN2C/2D-Selective Negative Allosteric Modulator of the N‑Methyl‑d‑aspartate Receptor.
저자
by
D'Erasmo, Michael P.
;
Akins, Nicholas S.
;
Ma, Peipei
;
Jing, Yao
;
Swanger, Sharon A.
, et al.
소스
ACS Chemical Neuroscience; 9/6/2023, Vol. 14 Issue 17, p3059-3076, 18p
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7 . Academic Journal
Alleviation of Cocaine Withdrawal and Pertinent Interactions between Salvinorin-Based Antagonists and Kappa Opioid Receptor.
저자
by
Akins, Nicholas S.
;
Salahuddin, Mohammed F.
;
Pandey, Pankaj
;
Kim, Seong Jong
;
Mahdi, Fakhri
, et al.
소스
ACS Chemical Neuroscience; 3/1/2023, Vol. 14 Issue 5, p958-976, 19p
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7 . Academic Journal
Novel GluN2B-Selective NMDA Receptor Negative Allosteric Modulator Possesses Intrinsic Analgesic Properties and Enhances Analgesia of Morphine in a Rodent Tail Flick Pain Model.
저자
by
Harris, Lynnea D.
;
Regan, Michael C.
;
Myers, Scott J.
;
Nocilla, Kelsey A.
;
Akins, Nicholas S.
, et al.
소스
ACS Chemical Neuroscience; 3/1/2023, Vol. 14 Issue 5, p917-935, 19p
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7 . Academic Journal
6,5‐Fused Ring, C2‐Salvinorin Ester, Dual Kappa and Mu Opioid Receptor Agonists as Analgesics Devoid of Anxiogenic Effects**.
저자
by
Akins, Nicholas S.
;
Mishra, Nisha
;
Harris, Hannah M.
;
Dudhipala, Narendar
;
Kim, Seong Jong
, et al.
소스
ChemMedChem; 4/5/2022, Vol. 17 Issue 7, p1-12, 12p
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7 . Academic Journal
Synthesis and Evaluation of Novel Tetrahydronaphthyridine CXCR4 Antagonists with Improved Drug-like Profiles.
저자
by
Jecs, Edgars
;
Tahirovic, Yesim A.
;
Wilson, Robert J.
;
Miller, Eric J.
;
Kim, Michelle
, et al.
소스
Journal of Medicinal Chemistry; 3/10/2022, Vol. 65 Issue 5, p4058-4084, 27p
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7 . Academic Journal
Allopregnanolone and neuroHIV: Potential benefits of neuroendocrine modulation in the era of antiretroviral therapy.
저자
by
Salahuddin, Mohammed F.
;
Qrareya, Alaa N.
;
Mahdi, Fakhri
;
Moss, Emaya
;
Akins, Nicholas S.
, et al.
소스
Journal of Neuroendocrinology
. Feb2022, Vol. 34 Issue 2, p1-15. 15p.
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7 . Academic Journal
Amino-Heterocycle Tetrahydroisoquinoline CXCR4 Antagonists with Improved ADME Profiles via Late-Stage Buchwald Couplings.
저자
by
Nguyen, Huy H.
;
Tahirovic, Yesim A.
;
Truax, Valarie M.
;
Wilson, Robert J.
;
Jecs, Edgars
, et al.
소스
ACS Medicinal Chemistry Letters; 10/14/2021, Vol. 12 Issue 10, p1605-1612, 8p
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