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1 .
Translational PK–PD for targeted protein degradation
저자
by
Derek W. Bartlett
;
Adam M. Gilbert
.
소스
Chemical Society Reviews
. 51:3477-3486
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4 .
Snapshots and ensembles of BTK and cIAP1 protein degrader ternary complexes
저자
by
Xidong Feng
;
Ye Che
;
Adam M. Gilbert
;
Reto Horst
;
Kris A. Borzilleri
, et al.
소스
Nature Chemical Biology
. 17:152-160
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7 .
Intramolecular Ring-Opening Decomposition of Aryl Azetidines
저자
by
Laura A. McAllister
;
Michael Aaron Brodney
;
Jane M. Withka
;
Jiangli Yan
;
Thomas N. O'Connell
, et al.
소스
ACS Med Chem Lett
Open Access (OpenAIRE)
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7 .
Inducing protein-protein interactions with molecular glues
저자
by
Adam M. Gilbert
;
Veerabahu Shanmugasundaram
;
Ye Che
;
Mark C. Noe
.
소스
Bioorganic & Medicinal Chemistry Letters
. 28:2585-2592
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6 . Academic Journal
(1-(4-(Naphthalen-2-yl)pyrimidin-2-yl)piperidin-4-yl)methanamine: A Wingless β-Catenin Agonist That Increases Bone Formation Rate.
저자
by
Jeffrey C. Pelletier
;
Joseph T. Lundquist
;
Adam M. Gilbert
;
Nipa Alon
;
Frederick J. Bex
, et al.
소스
Journal of Medicinal Chemistry
. Nov2009, Vol. 52 Issue 22, p6962-6965. 4p.
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7 .
Structure-Based Approach To Identify 5-[4-Hydroxyphenyl]pyrrole-2-carbonitrile Derivatives as Potent and Tissue Selective Androgen Receptor Modulators
저자
by
Christopher McNally
;
James J. Mousseau
;
Jay Wrobel
;
Carl Morris
;
Matthew R. Yudt
, et al.
소스
Journal of Medicinal Chemistry
. 60:6451-6457
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7 .
Clearance Prediction of Targeted Covalent Inhibitors by In Vitro-In Vivo Extrapolation of Hepatic and Extrahepatic Clearance Mechanisms
저자
by
Louis Leung
;
Justin I. Montgomery
;
Atli Thorarensen
;
Adam M. Gilbert
;
Timothy J. Strelevitz
, et al.
소스
Drug Metabolism and Disposition
. 45:1-7
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7 .
Optimization of a Dicarboxylic Series for in Vivo Inhibition of Citrate Transport by the Solute Carrier 13 (SLC13) Family
저자
by
Michael Herr
;
Daniel P. Canterbury
;
Derek M. Erion
;
Janice A. Brown
;
Mark Niosi
, et al.
소스
Journal of Medicinal Chemistry
. 59:1165-1175
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7 .
Intrinsic reactivity profile of electrophilic moieties to guide covalent drug design: N-α-acetyl-
l
-lysine as an amine nucleophile
저자
by
Jennifer A. Young
;
Mark Edward Flanagan
;
Jinshan M. Chen
;
Carmen N. Garcia-Irizarry
;
R. Scott Obach
, et al.
소스
MedChemComm
. 7:864-872
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7 .
Delineating the role of cooperativity in the design of potent PROTACs for BTK
저자
by
Suman Luthra
;
Graham M. West
;
Jeremy T. Starr
;
Matthew Frank Brown
;
Matthew F. Calabrese
, et al.
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