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1 . Academic Journal
Fragment merging approach for the design of thiazole/thiazolidine clubbed pyrazoline derivatives as anti-inflammatory agents: Synthesis, biopharmacological evaluation and molecular modeling studies
저자
by
Elgohary, Mohamed K.
;
Abd El Hadi, Soha R.
;
Abo-Ashour, Mahmoud F.
;
Abo-El Fetoh, Mohammed E.
;
Afify, Hassan
, et al.
소스
In
Bioorganic Chemistry
October 2023 139
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7 . Academic Journal
Novel benzenesulfonamides aryl and arylsulfone conjugates adopting tail/dual tail approaches: Synthesis, carbonic anhydrase inhibitory activity and molecular modeling studies
저자
by
Eldeeb, Assem H.
;
Abo-Ashour, Mahmoud F.
;
Angeli, Andrea
;
Bonardi, Alessandro
;
Lasheen, Deena S.
, et al.
소스
In
European Journal of Medicinal Chemistry
5 October 2021 221
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7 . Academic Journal
Identification of N-phenyl-2-(phenylsulfonyl)acetamides/propanamides as new SLC-0111 analogues: Synthesis and evaluation of the carbonic anhydrase inhibitory activities
저자
by
Elbadawi, Mostafa M.
;
Eldehna, Wagdy M.
;
Nocentini, Alessio
;
Abo-Ashour, Mahmoud F.
;
Elkaeed, Eslam B.
, et al.
소스
In
European Journal of Medicinal Chemistry
5 June 2021 218
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7 . Academic Journal
Development of isatin-thiazolo[3,2-a]benzimidazole hybrids as novel CDK2 inhibitors with potent in vitro apoptotic anti-proliferative activity: Synthesis, biological and molecular dynamics investigations
저자
by
Eldehna, Wagdy M.
;
El Hassab, Mahmoud A.
;
Abo-Ashour, Mahmoud F.
;
Al-Warhi, Tarfah
;
Elaasser, Mahmoud M.
, et al.
소스
In
Bioorganic Chemistry
May 2021 110
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7 . Academic Journal
3-Methylthiazolo[3,2-a]benzimidazole-benzenesulfonamide conjugates as novel carbonic anhydrase inhibitors endowed with anticancer activity: Design, synthesis, biological and molecular modeling studies
저자
by
Alkhaldi, Abdulsalam A.M.
;
Al-Sanea, Mohammad M.
;
Nocentini, Alessio
;
Eldehna, Wagdy M.
;
Elsayed, Zainab M.
, et al.
소스
In
European Journal of Medicinal Chemistry
1 December 2020 207
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7 . Academic Journal
3-Hydrazinoisatin-based benzenesulfonamides as novel carbonic anhydrase inhibitors endowed with anticancer activity: Synthesis, in vitro biological evaluation and in silico insights
저자
by
Abo-Ashour, Mahmoud F.
;
Eldehna, Wagdy M.
;
Nocentini, Alessio
;
Bonardi, Alessandro
;
Bua, Silvia
, et al.
소스
In
European Journal of Medicinal Chemistry
15 December 2019 184
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7 . Academic Journal
Enhancement of the tail hydrophobic interactions within the carbonic anhydrase IX active site via structural extension: Design and synthesis of novel N-substituted isatins-SLC-0111 hybrids as carbonic anhydrase inhibitors and antitumor agents
저자
by
Eldehna, Wagdy M.
;
Abo-Ashour, Mahmoud F.
;
Nocentini, Alessio
;
El-Haggar, Radwan S.
;
Bua, Silvia
, et al.
소스
In
European Journal of Medicinal Chemistry
15 January 2019 162:147-160
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7 . Academic Journal
Novel indole-thiazolidinone conjugates: Design, synthesis and whole-cell phenotypic evaluation as a novel class of antimicrobial agents
저자
by
Abo-Ashour, Mahmoud F.
;
Eldehna, Wagdy M.
;
George, Riham F.
;
Abdel-Aziz, Marwa M.
;
Elaasser, Mahmoud M.
, et al.
소스
In
European Journal of Medicinal Chemistry
5 December 2018 160:49-60
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7 . Academic Journal
Novel hydrazido benzenesulfonamides-isatin conjugates: Synthesis, carbonic anhydrase inhibitory activity and molecular modeling studies
저자
by
Abo-Ashour, Mahmoud F.
;
Eldehna, Wagdy M.
;
Nocentini, Alessio
;
Ibrahim, Hany S.
;
Bua, Silvia
, et al.
소스
In
European Journal of Medicinal Chemistry
5 September 2018 157:28-36
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7 . Academic Journal
Novel 4/3-((4-oxo-5-(2-oxoindolin-3-ylidene)thiazolidin-2-ylidene)amino) benzenesulfonamides: Synthesis, carbonic anhydrase inhibitory activity, anticancer activity and molecular modelling studies
저자
by
Eldehna, Wagdy M.
;
Abo-Ashour, Mahmoud F.
;
Nocentini, Alessio
;
Gratteri, Paola
;
Eissa, Ibrahim H.
, et al.
소스
In
European Journal of Medicinal Chemistry
20 October 2017 139:250-262
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