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1 . Academic Journal
Identification and optimisation of a pyrimidopyridone series of IRAK4 inhibitors
저자
by
Cumming, Iain A.
;
Degorce, Sébastien L.
;
Aagaard, Anna
;
Braybrooke, Erin L.
;
Davies, Nichola L.
, et al.
소스
In
Bioorganic & Medicinal Chemistry
1 June 2022 63
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7 . Academic Journal
Relocation of an internal proton donor in cytochrome c oxidase results in an altered p Ka and a non-integer pumping stoichiometry
저자
by
Gilderson, Gwen
;
Aagaard, Anna
;
Brzezinski, Peter
.
소스
In
Biophysical Chemistry
2002 98(1):105-114
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5 . Academic Journal
Fragment-Based Discovery of Novel Allosteric MEK1 Binders.
저자
by
Di Fruscia, Paolo
;
Edfeldt, Fredrik
;
Shamovsky, Igor
;
Collie, Gavin W.
;
Aagaard, Anna
, et al.
소스
ACS Medicinal Chemistry Letters; 2/11/2021, Vol. 12 Issue 2, p302-308, 7p
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7 . Periodical
AZD0284, a Potent, Selective, and Orally Bioavailable Inverse Agonist of Retinoic Acid Receptor-Related Orphan Receptor C2
저자
by
Narjes, Frank
;
Llinas, Antonio
;
von Berg, Stefan
;
Jirholt, Johan
;
Lever, Sarah
, et al.
소스
Journal of Medicinal Chemistry; September 2021, Vol. 64 Issue: 18 p13807-13829, 23p
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7 . Academic Journal
Synthesis and structure-activity relationship of 4-(1,3-benzothiazol-2-yl)-thiophene-2-sulfonamides as cyclin-dependent kinase 5 (cdk5)/p25 inhibitors
저자
by
Malmström, Jonas
;
Viklund, Jenny
;
Slivo, Can
;
Costa, Ana
;
Maudet, Mickaël
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 September 2012 22(18):5919-5923
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7 . Academic Journal
Discovery of Potent and Orally Bioavailable Inverse Agonists of the Retinoic Acid Receptor-Related Orphan Receptor C2.
저자
by
von Berg, Stefan
;
Xue, Yafeng
;
Collins, Mia
;
Llinas, Antonio
;
Olsson, Roine I.
, et al.
소스
ACS Medicinal Chemistry Letters; 2019, Vol. 10 Issue 6, p972-977, 6p
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7 . Academic Journal
Identification of Mineralocorticoid Receptor Modulators with Low Impact on Electrolyte Homeostasis but Maintained Organ Protection.
저자
by
Granberg, Kenneth L.
;
Yuan, Zhong-Qing
;
Lindmark, Bo
;
Edman, Karl
;
Kajanus, Johan
, et al.
소스
Journal of Medicinal Chemistry; 2/14/2019, Vol. 62 Issue 2, p1385-1406, 22p
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7 . Academic Journal
Potent and Orally Bioavailable Inverse Agonists of RORγt Resulting from Structure-Based Design.
저자
by
Narjes, Frank
;
Yafeng Xue
;
Stefan von Berg
;
Malmberg, Jesper
;
Llinas, Antonio
, et al.
소스
Journal of Medicinal Chemistry; 9/13/2018, Vol. 61 Issue 17, p7796-7813, 18p
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7 . Academic Journal
Structure and biophysical characterization of the human full-length neurturin-GFRa2 complex: A role for heparan sulfate in signaling.
저자
by
Sandmark, Jenny
;
Dahl, Göran
;
Öster, Linda
;
Bingze Xu
;
Johansson, Patrik
, et al.
소스
Journal of Biological Chemistry
. 4/13/2018, Vol. 293 Issue 15, p5492-5508. 17p.
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7 . Academic Journal
Preclinical pharmacology of AZD9977: A novel mineralocorticoid receptor modulator separating organ protection from effects on electrolyte excretion.
저자
by
Bamberg, Krister
;
Johansson, Ulrika
;
Edman, Karl
;
William-Olsson, Lena
;
Myhre, Susanna
, et al.
소스
PLoS ONE
. 2/23/2018, Vol. 13 Issue 2, p1-22. 22p.
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