Discovery and Optimization of an Azetidine Chemical Series As a Free Fatty Acid Receptor 2 (FFA2) Antagonist: From Hit to Clinic
- Resource Type
- Journal
- Authors
- Pizzonero, Mathieu; Dupont, Sonia; Babel, Marielle; Beaumont, Stephane; Bienvenu, Natacha; Blanque, Roland; Cherel, Laetitia; Christophe, Thierry; Crescenzi, Benedetta; De Lemos, Elsa; Delerive, Philippe; Deprez, Pierre; De Vos, Steve; Djata, Fatoumata; Fletcher, Stephen; Kopiejewski, Sabrina; L'Ebraly, Christelle; Lefrancois, Jean-Michel; Lavazais, Stephanie; Manioc, Murielle; Nelles, Luc; Oste, Line; Polancec, Denis; Quenehen, Vanessa; Soulas, Florilene; Triballeau, Nicolas; van der Aar, Ellen M.; Vandeghinste, Nick; Wakselman, Emanuelle; Brys, Reginald; Saniere, Laurent
- Source
- JOURNAL OF MEDICINAL CHEMISTRY; DEC 11 2014, 57 23, p10044-p10057, 14p.
- Subject
- Language
- English
- ISSN
- 15204804