Exploiting a water network to achieve enthalpy-driven, bromodomain-selective BET inhibitors
- Resource Type
- Article
- Authors
- Shadrick, William R.; Slavish, Peter J.; Chai, Sergio C.; Waddell, Brett; Connelly, Michele; Low, Jonathan A.; Tallant, Cynthia; Young, Brandon M.; Bharatham, Nagakumar; Knapp, Stefan; Boyd, Vincent A.; Morfouace, Marie; Roussel, Martine F.; Chen, Taosheng; Lee, Richard E.; Kiplin Guy, R.; Shelat, Anang A.; Potter, Philip M.
- Source
- In Bioorganic & Medicinal Chemistry 1 January 2018 26(1):25-36
- Subject
- Language
- ISSN
- 0968-0896