Discovery of 2-amino-3-amido-5-aryl-pyridines as highly potent, orally bioavailable, and efficacious PERK kinase inhibitors
- Resource Type
- Short Communication
- Authors
- Calvo, Veronica; Surguladze, David; Li, An-Hu; Surman, Matthew D.; Malibhatla, Srikanth; Bandaru, Madhavarao; Jonnalagadda, Suresh Krishna; Adarasandi, Ravi; Velmala, Madhusudhan; Singireddi, Durga Rama Prasad; Velpuri, Mahendar; Nareddy, Bhaskar Reddy; Sastry, Visweswara; Mandati, Chiranjeevi; Guguloth, Rambabu; Siddiqui, Shapi; Patil, Basanagoud S.; Chad, Elena; Wolfley, Jennifer; Gasparek, Jennifer; Feldman, Kirsten; Betzenhauser, Matthew; Wiens, Brent; Koszelak-Rosenblum, Mary; Zhu, Guangyu; Du, Hongwen; Rigby, Alan C.; Mulvihill, Mark J.
- Source
- In Bioorganic & Medicinal Chemistry Letters 1 July 2021 43
- Subject
- Language
- ISSN
- 0960-894X