Discovery of orally active butyrolactam 11β-HSD1 inhibitors
- Resource Type
- Source
- Bioorganic & Medicinal Chemistry Letters. 16:5555-5560
- Subject
Lactams Stereochemistry Clinical Biochemistry Administration, Oral Pharmaceutical Science Biochemistry Chemical synthesis Mice chemistry.chemical_compound Oral administration In vivo 11-beta-Hydroxysteroid Dehydrogenase Type 1 Drug Discovery Animals Humans Potency Molecular Biology Metabolic Syndrome chemistry.chemical_classification biology Chemistry Organic Chemistry Enzyme Enzyme inhibitor Lactam biology.protein Molecular Medicine Selectivity hormones, hormone substitutes, and hormone antagonists - Language
- ISSN
- 0960-894X