Discovery of (2R)-N-[3-[2-[(3-Methoxy-1-methyl-pyrazol-4-yl)amino]pyrimidin-4-yl]-1H-indol-7-yl]-2-(4-methylpiperazin-1-yl)propenamide (AZD4205) as a Potent and Selective Janus Kinase 1 Inhibitor
- Resource Type
- Source
- Journal of Medicinal Chemistry. 63:4517-4527
- Subject
0303 health sciences Janus Kinase 1 Inhibitor Chemistry Stereochemistry medicine.medical_treatment 01 natural sciences stat 0104 chemical sciences 010404 medicinal & biomolecular chemistry 03 medical and health sciences Cytokine Tyrosine kinase 2 Drug Discovery medicine Molecular Medicine Janus kinase 030304 developmental biology - Language
- ISSN
- 1520-4804
0022-2623