Synthesis and evaluation of substituted benzoisoquinolinones as potent inhibitors of Chk1 kinase
- Resource Type
- Source
- Bioorganic & Medicinal Chemistry Letters. 17:6280-6285
- Subject
Models, Molecular Photochemistry Stereochemistry Clinical Biochemistry Drug Evaluation, Preclinical Pharmaceutical Science Apoptosis Quinolones Crystallography, X-Ray Biochemistry Chemical synthesis Inhibitory Concentration 50 Structure-Activity Relationship chemistry.chemical_compound Residue (chemistry) Cell Line, Tumor Drug Discovery Humans Transferase Structure–activity relationship Enzyme Inhibitors Molecular Biology chemistry.chemical_classification Binding Sites Molecular Structure biology Organic Chemistry Enzyme chemistry Enzyme inhibitor Checkpoint Kinase 1 Lactam biology.protein Molecular Medicine Amine gas treating Protein Kinases - Language
- ISSN
- 0960-894X