In vitro modulation of multidrug resistance by pregnane steroids and in vivo inhibition of tumour development by 7α-OBz-11α(R)-OTHP-5β-pregnanedione in K562/R7 and H295R cell xenografts
- Resource Type
- Source
- Journal of Enzyme Inhibition and Medicinal Chemistry
Journal of Enzyme Inhibition and Medicinal Chemistry, Informa Healthcare, 2019, 34 (1), pp.684-691. ⟨10.1080/14756366.2019.1575825⟩
Journal of Enzyme Inhibition and Medicinal Chemistry, 2019, 34 (1), pp.684-691. ⟨10.1080/14756366.2019.1575825⟩
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 34, Iss 1, Pp 684-691 (2019) - Subject
Cell Molecular Conformation Mice, SCID [CHIM.THER]Chemical Sciences/Medicinal Chemistry Multidrug resistance 01 natural sciences Mice chemistry.chemical_compound pregnane modulators Drug Discovery Tumor Cells, Cultured Adrenocortical carcinoma P-glycoprotein biology Pregnane General Medicine Pregnanes Drug Resistance, Multiple 3. Good health medicine.anatomical_structure xenografts [SDV.SP.PHARMA] Life Sciences [q-bio]/Pharmaceutical sciences/Pharmacology Female Research Paper medicine.drug [SDV.SP.MED] Life Sciences [q-bio]/Pharmaceutical sciences/Medication Cell Survival [CHIM.THER] Chemical Sciences/Medicinal Chemistry Antineoplastic Agents non-steroidogenic and steroidogenic cell lines Structure-Activity Relationship [SDV.SP.MED]Life Sciences [q-bio]/Pharmaceutical sciences/Medication In vivo medicine Animals Humans Doxorubicin Cell Proliferation Pharmacology Dose-Response Relationship, Drug 010405 organic chemistry lcsh:RM1-950 Neoplasms, Experimental medicine.disease In vitro 0104 chemical sciences 010404 medicinal & biomolecular chemistry lcsh:Therapeutics. Pharmacology chemistry Drug Resistance, Neoplasm Cell culture biology.protein Cancer research [SDV.SP.PHARMA]Life Sciences [q-bio]/Pharmaceutical sciences/Pharmacology Drug Screening Assays, Antitumor - Language
- English
- ISSN
- 1475-6366
1475-6374