Discovery and optimization of imidazo[1,2-a]pyridine inhibitors of insulin-like growth factor-1 receptor (IGF-1R)
- Resource Type
- Source
- Bioorganic & Medicinal Chemistry Letters. 19:1004-1008
- Subject
Pyridines Chemistry, Pharmaceutical medicine.medical_treatment Clinical Biochemistry Molecular Conformation Administration, Oral Pharmaceutical Science Crystallography, X-Ray Biochemistry Receptor, IGF Type 1 Inhibitory Concentration 50 Mice Insulin-like growth factor Growth factor receptor In vivo Cell Line, Tumor Drug Discovery medicine Animals Humans Receptor Molecular Biology Insulin-like growth factor 1 receptor Aniline Compounds biology Chemistry Organic Chemistry Receptor, Insulin In vitro Insulin receptor Models, Chemical Enzyme inhibitor Drug Design biology.protein Molecular Medicine - Language
- ISSN
- 0960-894X