Identification of diamino chromone-2-carboxamides as MCHr1 antagonists with minimal hERG channel activity
- Resource Type
- Source
- Bioorganicmedicinal chemistry letters. 17(8)
- Subject
Patch-Clamp Techniques medicine.drug_class Stereochemistry Clinical Biochemistry hERG Pharmaceutical Science Carboxamide Biochemistry Chemical synthesis chemistry.chemical_compound Inhibitory Concentration 50 Mice In vivo Drug Discovery medicine Animals Humans Pharmacokinetics Patch clamp Obesity Receptors, Pituitary Hormone Molecular Biology biology Organic Chemistry Amides In vitro Ether-A-Go-Go Potassium Channels chemistry Hormone receptor Chromones Chromone biology.protein Molecular Medicine - Language
- ISSN
- 0960-894X