Discovery of novel quinoline sulphonamide derivatives as potent, selective and orally active RORγ inverse agonists
- Resource Type
- Short Communication
- Authors
- Amaudrut, Jérôme; Argiriadi, Maria A.; Barth, Martine; Breinlinger, Eric C.; Bressac, Didier; Broqua, Pierre; Calderwood, David J.; Chatar, Mohamed; Cusack, Kevin P.; Gauld, Stephen B.; Jacquet, Sébastien; Kamath, Rajesh V.; Kort, Michael E.; Lepais, Valérie; Luccarini, Jean-Michel; Masson, Philippe; Montalbetti, Christian; Mounier, Laurent; Potin, Dominique; Poupardin, Olivia; Rouaud, Sylvie; Spitzer, Luc; Wallace, Craig D.
- Source
- In Bioorganic & Medicinal Chemistry Letters 15 July 2019 29(14):1799-1806
- Subject
- Language
- ISSN
- 0960-894X