Unexpected equivalent potency of a constrained chromene enantiomeric pair rationalized by co-crystal structures in complex with estrogen receptor alpha
Resource Type
Short Communication
Authors
Zhang, Birong ; Kiefer, James R. ; Blake, Robert A. ; Chang, Jae H. ; Hartman, Steven ; Ingalla, Ellen Rei ; Kleinheinz, Tracy ; Mody, Vidhi ; Nannini, Michelle ; Ortwine, Daniel F. ; Ran, Yingqing ; Sambrone, Amy ; Sampath, Deepak ; Vinogradova, Maia ; Zhong, Yu ; Nwachukwu, Jerome C. ; Nettles, Kendall W. ; Lai, Tommy ; Liao, Jiangpeng ; Zheng, Xiaoping ; Chen, Hai ; Wang, Xiaojing ; Liang, Jun
Source
In Bioorganic & Medicinal Chemistry Letters 1 April 2019 29(7):905-911
Subject
Language
ISSN
0960-894X