Hydroxyethylamine-based inhibitors of BACE1: P1–P3 macrocyclization can improve potency, selectivity, and cell activity
- Resource Type
- Short Communication
- Authors
- Pennington, Lewis D.; Whittington, Douglas A.; Bartberger, Michael D.; Jordan, Steven R.; Monenschein, Holger; Nguyen, Thomas T.; Yang, Bryant H.; Xue, Qiufen M.; Vounatsos, Filisaty; Wahl, Robert C.; Chen, Kui; Wood, Stephen; Citron, Martin; Patel, Vinod F.; Hitchcock, Stephen A.; Zhong, Wenge
- Source
- In Bioorganic & Medicinal Chemistry Letters 1 August 2013 23(15):4459-4464
- Subject
- Language
- ISSN
- 0960-894X