Discovery of a Potent and Orally Bioavailable Zwitterionic Series of Selective Estrogen Receptor Degrader-Antagonists.
- Resource Type
- Article
- Authors
- Scott, James S.; Stead, Darren; Barlaam, Bernard; Breed, Jason; Carbajo, Rodrigo J.; Chiarparin, Elisabetta; Cureton, Natalie; Davey, Paul R. J.; Fisher, David I.; Gangl, Eric T.; Grebe, Tyler; Greenwood, Ryan D.; Hande, Sudhir; Hatoum-Mokdad, Holia; Hughes, Samantha J.; Hunt, Thomas A.; Johnson, Tony; Kavanagh, Stefan L.; Klinowska, Teresa C. M.; Larner, Carrie J. B.
- Source
- Journal of Medicinal Chemistry; 2/23/2023, Vol. 66 Issue 4, p2918-2945, 28p
- Subject
- Language
- ISSN
- 00222623