Size-Reduced Macrocyclic Analogues of [Pyr¹]-apelin-13 Showing Negative Gα12 Bias Still Produce Prolonged Cardiac Effects.
- Resource Type
- Article
- Authors
- Tran, Kien; Sainsily, Xavier; Côté, Jérôme; Coquerel, David; Couvineau, Pierre; Saibi, Sabrina; Haroune, Lounès; Besserer-Offroy, Élie; Flynn-Robitaille, Joël; Rojas, Martin Resua; Murza, Alexandre; Longpré, Jean-Michel; Auger-Messier, Mannix; Lesur, Olivier; Bouvier, Michel; Marsault, Éric; Boudreault, Pierre-Luc; Sarret, Philippe
- Source
- Journal of Medicinal Chemistry; 1/13/2022, Vol. 65 Issue 1, p531-551, 21p
- Subject
- Language
- ISSN
- 00222623