Design of Conformationally Constrained Acyl Sulfonamide Isosteres: Identification of N-([1,2,4]Triazolo[4,3-a]pyridin-3-yl)methane-sulfonamidesas Potent and Selective hNa(v)1.7 Inhibitors for the Treatment of Pain
Resource Type
Journal
Authors
Focken, Thilo ; Chowdhury, Sultan ; Zenova, Alla ; Grimwood, Michael E. ; Chabot, Christine ; Sheng, Tao ; Hemeon, Ivan ; Decker, Shannon M. ; Wilson, Michael ; Bichler, Paul ; Jia, Qi ; Sun, Shaoyi ; Young, Clint ; Lin, Sophia ; Goodchild, Samuel J. ; Shuart, Noah G. ; Chang, Elaine ; Xie, Zhiwei ; Li, Bowen ; Khakh, Kuldip ; Bankar, Girish ; Waldbrook, Matthew ; Kwan, Rainbow ; Nelkenbrecher, Karen ; Tari, Parisa Karimi ; Chahal, Navjot ; Sojo, Luis ; Robinette, C. Lee ; White, Andrew D. ; Chen, Chien-An ; Zhang, Yi ; Pang, Jodie ; Chang, Jae H. ; Hackos, David H. ; Johnson, J. P. ; Cohen, Charles J. ; Ortwine, Daniel F. ; Sutherlin, Daniel P. ; Dehnhardt, Christoph M. ; Safina, Brian S.
Source
JOURNAL OF MEDICINAL CHEMISTRY ; JUN 14 2018, 61 11, p4810-p4831, 22p.
Subject
Language
English
ISSN
15204804