Discovery of APD334: Design of a Clinical Stage Functional Antagonist of the Sphingosine-1-phosphate-1 Receptor
- Resource Type
- Journal
- Authors
- Buzard, Daniel J.; Kim, Sun Hee; Lopez, Luis; Kawasaki, Andrew; Zhu, Xiuwen; Moody, Jeanne; Thoresen, Lars; Calderon, Imelda; Ullman, Brett; Han, Sangdon; Lehmann, Juerg; Gharbaoui, Tawfik; Sengupta, Dipanjan; Calvano, Lorene; Montalban, Antonio Garrido; Ma, You-An; Sage, Carleton; Gao, Yinghong; Semple, Graeme; Edwards, Jeff; Barden, Jeremy; Morgan, Michael; Chen, Weichao; Usmani, Khawja; Chen, Chuan; Sadeque, Abu; Christopher, Ronald J.; Thatte, Jayant; Fu, Lixia; Solomon, Michelle; Mills, David; Whelan, Kevin; Al-Shamma, Hussien; Gatlin, Joel; Minh Le; Gaidarov, Ibragim; Anthony, Todd; Unett, David J.; Blackburn, Anthony; Rueter, Jaimie; Stirn, Scott; Behan, Dominic P.; Jones, Robert M.
- Source
- ACS MEDICINAL CHEMISTRY LETTERS; DEC 2014, 5 12, p1313-p1317, 5p.
- Subject
- Language
- English
- ISSN
- 19485875