Synthesis of BACE Inhibitor LY2886721. Part II. Isoxazolidines as Precursors to Chiral Aminothiazines, Selective Peptide Coupling, and a Controlled Reactive Crystallization
Resource Type
Journal
Authors
Hansen, Marvin M. ; Jarmer, Daniel J. ; Arslantas, Enver ; DeBaillie, Amy C. ; Frederick, Andrea L. ; Harding, Molly ; Hoard, David W. ; Hollister, Adrienne ; Huber, Dominique ; Kolis, Stanley P. ; Kuehne-Willmore, Jennifer E. ; Kull, Thomas ; Laurila, Michael E. ; Linder, Ryan J. ; Martin, Thomas J. ; Martinelli, Joseph R. ; McCulley, Michael J. ; Richey, Rachel N. ; Starkey, Derek R. ; Ward, Jeffrey A. ; Zaborenko, Nikolay ; Zweifel, Theo
Source
ORGANIC PROCESS RESEARCH & DEVELOPMENT ; SEP 2015, 19 9, p1214-p1230, 17p.
Subject
Language
English
ISSN
1520586X