Discovery of Novel Dot1L Inhibitors through a Structure-Based Fragmentation Approach
- Resource Type
- Journal
- Authors
- Chen, Chao; Zhu, Hugh; Stauffer, Frederic; Caravatti, Giorgio; Vollmer, Susanne; Machauer, Rainer; Holzer, Philipp; Mobitz, Henrik; Scheufler, Clemens; Klumpp, Martin; Tiedt, Ralph; Beyer, Kim S.; Calkins, Keith; Guthy, Daniel; Kiffe, Michael; Zhang, Jeff; Gaul, Christoph
- Source
- ACS MEDICINAL CHEMISTRY LETTERS; AUG 2016, 7 8, p735-p740, 6p.
- Subject
- Language
- English
- ISSN
- 19485875