4-(3-Trifluoromethylphenyl)-pyrimidine-2-carbonitrile as cathepsin S inhibitors: N3, not N1 is critically important
- Resource Type
- Short Communication
- Authors
- Cai, Jiaqiang; Fradera, Xavier; van Zeeland, Mario; Dempster, Maureen; Cameron, Kenneth S.; Bennett, D. Jonathan; Robinson, John; Popplestone, Lucy; Baugh, Mark; Westwood, Paul; Bruin, John; Hamilton, William; Kinghorn, Emma; Long, Clive; Uitdehaag, Joost C.M.
- Source
- In Bioorganic & Medicinal Chemistry Letters 1 August 2010 20(15):4507-4510
- Subject
- Language
- ISSN
- 0960-894X