Structure-based optimization of hydroxylactam as potent, cell-active inhibitors of lactate dehydrogenase
- Resource Type
- Short Communication
- Authors
- Wei, BinQing; Robarge, Kirk; Labadie, Sharada S.; Chen, Jinhua; Corson, Laura B.; DiPasquale, Antonio; Dragovich, Peter S.; Eigenbrot, Charles; Evangelista, Marie; Fauber, Benjamin P.; Hitz, Anna; Hong, Rebecca; Lai, Kwong Wah; Liu, Wenfeng; Ma, Shuguang; Malek, Shiva; O'Brien, Thomas; Pang, Jodie; Peterson, David; Salphati, Laurent; Sampath, Deepak; Sideris, Steven; Ultsch, Mark; Xu, Zijin; Yen, Ivana; Yu, Dong; Yue, Qin; Zhou, Aihe; Purkey, Hans E.
- Source
- In Bioorganic & Medicinal Chemistry Letters 1 March 2022 59
- Subject
- Language
- ISSN
- 0960-894X