Kinesin spindle protein (KSP) inhibitors. Part 7: Design and synthesis of 3,3-disubstituted dihydropyrazolobenzoxazines as potent inhibitors of the mitotic kinesin KSP
- Resource Type
- Source
- Bioorganic & Medicinal Chemistry Letters. 17:5671-5676
- Subject
Stereochemistry medicine.drug_class Clinical Biochemistry Kinesins Mitosis Pharmaceutical Science Carboxamide Biochemistry Chemical synthesis Cell Line Structure-Activity Relationship Dogs In vivo Drug Discovery medicine Animals Humans Molecular Biology chemistry.chemical_classification Molecular Structure biology Organic Chemistry Benzoxazines Spindle apparatus Enzyme chemistry Enzyme inhibitor Drug Design biology.protein Pyrazoles Molecular Medicine Kinesin Hydrogen - Language
- ISSN
- 0960-894X