Structural basis of CXC chemokine receptor 2 activation and signalling
- Resource Type
- Authors
- Kaiwen, Liu; Lijie, Wu; Shuguang, Yuan; Meng, Wu; Yueming, Xu; Qianqian, Sun; Shu, Li; Suwen, Zhao; Tian, Hua; Zhi-Jie, Liu
- Source
- Nature. 585(7823)
- Subject
- Models, Molecular
Structure-Activity Relationship
Allosteric Regulation
Interleukin-8
Humans
Chemokines
GTP-Binding Protein alpha Subunits, Gi-Go
Allosteric Site
Receptors, Interleukin-8B
Protein Binding
Signal Transduction
Substrate Specificity
- Language
- ISSN
- 1476-4687
Chemokines and their receptors mediate cell migration, which influences multiple fundamental biological processes and disease conditions such as inflammation and cancer