Discovery of 1H-Pyrazol-3(2H)-ones as Potent and Selective Inhibitors of Protein Kinase R-like Endoplasmic Reticulum Kinase (PERK)
- Resource Type
- Source
- Journal of Medicinal Chemistry. 58:1426-1441
- Subject
Models, Molecular endocrine system Dose-Response Relationship, Drug Molecular Structure Kinase Drug discovery Chemistry Endoplasmic reticulum Mice, Nude Protein kinase R In vitro Mice Structure-Activity Relationship eIF-2 Kinase Biochemistry In vivo Drug Discovery Animals Humans Pyrazoles Molecular Medicine Structure–activity relationship PERK inhibitors Protein Kinase Inhibitors Cells, Cultured - Language
- ISSN
- 1520-4804
0022-2623