Discovery of a novel series of guanidinebenzoates as gut-restricted enteropeptidase and trypsin dual inhibitors for the treatment of metabolic syndrome
- Resource Type
- Source
- Bioorganicmedicinal chemistry letters. 40
- Subject
Enteropeptidase Trypsin inhibitor Clinical Biochemistry Pharmaceutical Science CHO Cells Diet, High-Fat 01 natural sciences Biochemistry Benzoates Guanidines Feces Structure-Activity Relationship Cricetulus Drug Discovery Aqueous solubility medicine Animals Humans Obesity Molecular Biology Metabolic Syndrome Molecular Structure 010405 organic chemistry Chemistry Organic Chemistry Proteins medicine.disease Trypsin 0104 chemical sciences Bioavailability Protein excretion Mice, Inbred C57BL 010404 medicinal & biomolecular chemistry Molecular Medicine Cattle Metabolic syndrome Trypsin Inhibitors medicine.drug - Language
- ISSN
- 1464-3405