Discovery of Clinical Candidate CHF-6366: A Novel Super-soft Dual Pharmacology Muscarinic Antagonist and β
- Resource Type
- Authors
- Laura, Carzaniga; Ian D, Linney; Andrea, Rizzi; Maurizio, Delcanale; Wolfgang, Schmidt; Christopher K, Knight; Fiorella, Pastore; Daniela, Miglietta; Chiara, Carnini; Nicola, Cesari; Benedetta, Riccardi; Valentina, Mileo; Luca, Venturi; Elisa, Moretti; Wesley P, Blackaby; Riccardo, Patacchini; Alessandro, Accetta; Matteo, Biagetti; Franco, Bassani; Marina, Tondelli; Annalisa, Murgo; Loredana, Battipaglia; Gino, Villetti; Paola, Puccini; Silvia, Catinella; Maurizio, Civelli; Fabio, Rancati
- Source
- Journal of medicinal chemistry. 65(15)
- Subject
- Pulmonary Disease, Chronic Obstructive
Administration, Inhalation
Drug Discovery
Humans
Muscarinic Antagonists
Adrenergic beta-2 Receptor Agonists
Lung
Bronchodilator Agents
- Language
- ISSN
- 1520-4804
The development of molecules embedding two distinct pharmacophores acting as muscarinic antagonists and β