Driving Potency with Rotationally Stable Atropisomers: Discovery of Pyridopyrimidinedione-Carbazole Inhibitors of BTK.
- Resource Type
- Article
- Authors
- Srivastava, Anurag S.; Ko, Soo; Watterson, Scott H.; Pattoli, Mark A.; Skala, Stacey; Cheng, Lihong; Obermeier, Mary T.; Vickery, Rodney; Discenza, Lorell N.; D'Arienzo, Celia J.; Gillooly, Kathleen M.; Taylor, Tracy L.; Pulicicchio, Claudine; McIntyre, Kim W.; Yip, Shiuhang; Li, Peng; Sun, Dawn; Wu, Dauh-Rurng; Dai, Jun; Wang, Chunlei
- Source
- ACS Medicinal Chemistry Letters; 11/12/2020, Vol. 11 Issue 11, p2195-2203, 9p
- Subject
- Language
- ISSN
- 19485875