Peptidomimetic α-Acyloxymethylketone Warheads with Six-Membered Lactam P1 Glutamine Mimic: SARS-CoV-2 3CL Protease Inhibition, Coronavirus Antiviral Activity, and in Vitro Biological Stability.
- Resource Type
- Article
- Authors
- Bing Bai; Belovodskiy, Alexandr; Hena, Mostofa; Kandadai, Appan Srinivas; Joyce, Michael A.; Saffran, Holly A.; Shields, Justin A.; Khan, Muhammad Bashir; Arutyunova, Elena; Jimmy Lu; Bajwa, Sardeev K.; Hockman, Darren; Fischer, Conrad; Lamer, Tess; Vuong, Wayne; van Belkum, Marco J.; Zhengxian Gu; Fusen Lin; Yanhua Du; Jia Xu
- Source
- Journal of Medicinal Chemistry; 2/24/2022, Vol. 65 Issue 4, p2905-2925, 21p
- Subject
- Language
- ISSN
- 00222623