Optimization of Selectivity and Pharmacokinetic Properties of Salt‑Inducible Kinase Inhibitors that Led to the Discovery of Pan-SIK Inhibitor GLPG3312.
Resource Type
Article
Authors
Temal-Laib, Taouès ; Peixoto, Christophe ; Desroy, Nicolas ; De Lemos, Elsa ; Bonnaterre, Florence ; Bienvenu, Natacha ; Picolet, Olivier ; Sartori, Eric ; Bucher, Denis ; López-Ramos, Miriam ; Roca Magadán, Carlos ; Laenen, Wendy ; Flower, Thomas ; Mollat, Patrick ; Bugaud, Olivier ; Touitou, Robert ; Pereira Fernandes, Anna ; Lavazais, Stephanie ; Monjardet, Alain ; Borgonovi, Monica
Source
Journal of Medicinal Chemistry; 1/11/2024, Vol. 67 Issue 1, p380-401, 22p
Subject
Language
ISSN
00222623