Discovery of GLPG1972/S201086, a Potent, Selective, and Orally Bioavailable ADAMTS‑5 Inhibitor for the Treatment of Osteoarthritis.
- Resource Type
- Article
- Authors
- Brebion, Franck; Gosmini, Romain; Deprez, Pierre; Varin, Marie; Peixoto, Christophe; Alvey, Luke; Jary, Hélène; Bienvenu, Natacha; Triballeau, Nicolas; Blanque, Roland; Cottereaux, Céline; Christophe, Thierry; Vandervoort, Nele; Mollat, Patrick; Touitou, Robert; Leonard, Philip; Ceuninck, Frédéric De; Botez, Iuliana; Monjardet, Alain; van der Aar, Ellen
- Source
- Journal of Medicinal Chemistry; 3/25/2021, Vol. 64 Issue 6, p2937-2952, 16p
- Subject
- Language
- ISSN
- 00222623