Picomolar FKBP inhibitors enabled by a single water-displacing methyl group in bicyclic [4.3.1] aza-amides.
- Resource Type
- Article
- Authors
- Kolos, Jürgen M.; Pomplun, Sebastian; Sascha Jung; Rieß, Benedikt; Purder, Patrick L.; Voll, Andreas M.; Merz, Stephanie; Gnatzy, Monika; Geiger, Thomas M.; Quist-Løkken, Ingrid; Jatzlau, Jerome; Knaus, Petra; Holien, Toril; Bracher, Andreas; Meyners, Christian; Czodrowski, Paul; Krewald, Vera; Hausch, Felix
- Source
- Chemical Science; 11/28/2021, Vol. 12 Issue 44, p14758-14765, 8p
- Subject
- Language
- ISSN
- 20416520