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1 . Academic Journal
Targeted kinase degradation via the KLHDC2 ubiquitin E3 ligase
저자
by
Kim, Younghoon
;
Seo, Pooreum
;
Jeon, Eunhye
;
You, Inchul
;
Hwang, Kyubin
, et al.
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Cell Chemical Biology
16 November 2023 30(11):1414-1420
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7 . Academic Journal
The rise of degrader drugs
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Teng, Mingxing
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Gray, Nathanael S.
.
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Cell Chemical Biology
17 August 2023 30(8):864-878
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4 . Academic Journal
New scaffolds for type II JAK2 inhibitors overcome the acquired G993A resistance mutation
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by
Arwood, Matthew L.
;
Liu, Yao
;
Harkins, Shannon K.
;
Weinstock, David M.
;
Yang, Lei
, et al.
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Cell Chemical Biology
15 June 2023 30(6):618-631
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7 . Academic Journal
CDK7 controls E2F- and MYC-driven proliferative and metabolic vulnerabilities in multiple myeloma
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by
Yao, Yao
;
Ng, Jessica Fong
;
Park, Woojun Daniel
;
Samur, Mehmet
;
Morelli, Eugenio
, et al.
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Blood
8 June 2023 141(23):2841-2852
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7 . Academic Journal
USP9X mediates an acute adaptive response to MAPK suppression in pancreatic cancer but creates multiple actionable therapeutic vulnerabilities
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by
Perurena, Naiara
;
Lock, Rebecca
;
Davis, Rachel A.
;
Raghavan, Srivatsan
;
Pilla, Natalie F.
, et al.
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Cell Reports Medicine
18 April 2023 4(4)
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7 . Academic Journal
Development of potent and selective degraders of PI5P4Kγ
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by
Ji, Wenzhi
;
Wang, Eric S.
;
Manz, Theresa D.
;
Jiang, Jie
;
Donovan, Katherine A.
, et al.
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European Journal of Medicinal Chemistry
5 February 2023 247
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7 . Academic Journal
Exploring the target scope of KEAP1 E3 ligase-based PROTACs
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by
Du, Guangyan
;
Jiang, Jie
;
Henning, Nathaniel J.
;
Safaee, Nozhat
;
Koide, Eriko
, et al.
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Cell Chemical Biology
20 October 2022 29(10):1470-1481
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7 . Academic Journal
Temporal resolution of gene derepression and proteome changes upon PROTAC-mediated degradation of BCL11A protein in erythroid cells
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Mehta, Stuti
;
Buyanbat, Altantsetseg
;
Kai, Yan
;
Karayel, Ozge
;
Goldman, Seth Raphael
, et al.
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Cell Chemical Biology
18 August 2022 29(8):1273-1287
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7 . Academic Journal
Synthesis and Structure–Activity relationships of cyclin-dependent kinase 11 inhibitors based on a diaminothiazole scaffold
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by
Li, Zhengnian
;
Ishida, Ryosuke
;
Liu, Yan
;
Wang, Jinhua
;
Li, Yina
, et al.
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European Journal of Medicinal Chemistry
5 August 2022 238
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7 . Academic Journal
Structure-activity relationship study of THZ531 derivatives enables the discovery of BSJ-01-175 as a dual CDK12/13 covalent inhibitor with efficacy in Ewing sarcoma
저자
by
Jiang, Baishan
;
Jiang, Jie
;
Kaltheuner, Ines H.
;
Iniguez, Amanda Balboni
;
Anand, Kanchan
, et al.
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European Journal of Medicinal Chemistry
5 October 2021 221
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