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1 . Academic Journal
Discovery of E2730, a novel selective uncompetitive GAT1 inhibitor, as a candidate for anti‐seizure medication
저자
by
Kazuyuki Fukushima
;
Hiroyuki Higashiyama
;
Yuji Kazuta
;
Keisuke Hashimoto
;
Naoto Watanabe
, et al.
소스
Epilepsia Open, Vol 8, Iss 3, Pp 834-845 (2023)
Open Access (Wiley)
Open Access (DOAJ)
Web of Science
Scopus
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7 . Academic Journal
Discovery of a novel and potent dual orexin 1/2 receptor antagonist, lemborexant (E2006), for the treatment of sleep disorders / 睡眠障害治療薬を志向したオレキシン1/2受容体新規デュアルアンタゴニストlemborexant(E2006)の創製
저자
by
Carsten Beuckmann
;
Taro Terauchi
;
Yoshimitsu Naoe
;
Yu Yoshida
;
Yuji Kazuta
, et al.
소스
MEDCHEM NEWS. 2019, 29(2):69
Find it @ DONGA
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7 . Academic Journal
P-253 DEVELOPMENT OF POTENT HISTAMINE H_3 AND/OR H_4 RECEPTOR ANTAGONISTS BY THE STEREOCHEMICAL DIVERSITY-ORIENTED CONFORMATIONAL RESTRICTION STRATEGY
저자
by
Akira Matsuda
;
Hideki Hayashi
;
Mizuki Watanabe
;
Satoshi Shuto
;
Shizuo Yamada
, et al.
소스
International Symposium on the Chemistry of Natural Products. 2006, 253
Open Access (JSTAGE)
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7 .
Discovery of
E2730
, a novel selective uncompetitive
GAT1
inhibitor, as a candidate for anti‐seizure medication
저자
by
Kazuyuki Fukushima
;
Hiroyuki Higashiyama
;
Yuji Kazuta
;
Keisuke Hashimoto
;
Naoto Watanabe
, et al.
소스
Epilepsia Open
.
Open Access (OpenAIRE)
Scopus
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Export
E-Mail
EndNote
RefWorks
7 .
Silinanyl Rhodamines and Silinanyl Fluoresceins for Super-Resolution Microscopy
저자
by
Masatoshi Suganuma
;
Masaya Okada
;
Yuji Kazuta
;
Kazuto Yamashita
;
Shingo Fujiyama
, et al.
소스
The Journal of Physical Chemistry B
. 125:8703-8711
Web of Science
Scopus
JCR 저널정보
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7 .
Design, synthesis, and structure–activity relationships of a series of novel N-aryl-2-phenylcyclopropanecarboxamide that are potent and orally active orexin receptor antagonists
저자
by
Carsten T. Beuckmann
;
Yuji Kazuta
;
Osamu Takenaka
;
Fumihiro Ozaki
;
Yu Yoshida
, et al.
소스
Bioorganic & Medicinal Chemistry
. 22:6071-6088
Web of Science
Scopus
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7 .
Stereochemical Diversity-Oriented Conformational Restriction Strategy. Development of Potent Histamine H3 and/or H4 Receptor Antagonists with an Imidazolylcyclopropane Structure
저자
by
and Akira Matsuda
;
Yuji Kazuta
;
Mizuki Watanabe
;
Shizuo Yamada
;
Hideki Hayashi
, et al.
소스
Journal of Medicinal Chemistry
. 49:5587-5596
Web of Science
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7 .
Highly Stereoselective Grignard Addition to Cis-Substituted C-Cyclopropylaldonitrones. The Bisected s-Trans Transition State Can Be Stabilized Effectively by the Lewis Acid-Coordination
저자
by
Satoshi Shuto
;
and Akira Matsuda
;
Hiroshi Abe
;
Yuji Kazuta
.
소스
The Journal of Organic Chemistry
. 69:9143-9150
Web of Science
Scopus
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6 .
The unusual 1,4-chelation-controlled nucleophilic addition to aldehydes with high stereoselectivity. A systematic study of stereoselectivity in the addition reaction of carbon nucleophiles to cis-substituted cyclopropanecarbaldehydes
저자
by
Akira Matsuda
;
Hiroshi Abe
;
Yuji Kazuta
;
Satoshi Shuto
;
Tamotsu Yamamoto
.
소스
Tetrahedron
. 60:6689-6703
Web of Science
Scopus
JCR 저널정보
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7 .
Cyclopropane-Based Conformational Restriction of Histamine. (1S,2S)-2-(2-Aminoethyl)-1-(1H-imidazol-4-yl)cyclopropane, a Highly Selective Agonist for the Histamine H3 Receptor, Having a cis-Cyclopropane Structure
저자
by
and Akira Matsuda
;
Kentaro Natsume
;
Kazufumi Hirano
;
Kiyoshi Furuichi
;
§ Shun-ichiro Matsumoto
, et al.
소스
Journal of Medicinal Chemistry
. 46:1980-1988
Web of Science
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