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1 . Academic Journal
New evolutions in the BACE1 inhibitor field from 2014 to 2018
저자
by
Hsiao, Chien-Chi
;
Rombouts, Frederik
;
Gijsen, Harrie J.M.
.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 March 2019 29(6):761-777
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5 . Academic Journal
3,3-Difluoro-3,4,5,6-tetrahydropyridin-2-amines: Potent and permeable BACE-1 inhibitors
저자
by
Peschiulli, Aldo
;
Oehlrich, Daniel
;
Rombouts, Frederik
;
Vos, Ann
;
Gijsen, Harrie JM
.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 April 2020 30(8)
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7 . Academic Journal
Expedient Access to Cyanated N‐Heterocycles by Direct Flow‐Electrochemical C(sp
2
)−H Activation.
저자
by
Carvalho, Mary‐Ambre
;
Demin, Samuël
;
Martinez‐Lamenca, Carolina
;
Romanov‐Michailidis, Fedor
;
Lam, Kevin
, et al.
소스
Chemistry - A European Journal
. 1/3/2022, Vol. 28 Issue 1, p1-6. 6p.
Full Text (Wiley)
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7 . Academic Journal
Anilinotriazoles as potent gamma secretase modulators
저자
by
Velter, Adriana I.
;
Bischoff, François P.
;
Berthelot, Didier
;
De Cleyn, Michel
;
Oehlrich, Daniel
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 December 2014 24(24):5805-5813
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7 . Academic Journal
Discovery of a new series of [1,2,4]triazolo[4,3-a]quinoxalines as dual phosphodiesterase 2/phosphodiesterase 10 (PDE2/PDE10) inhibitors
저자
by
Andrés, José-Ignacio
;
Buijnsters, Peter
;
De Angelis, Meri
;
Langlois, Xavier
;
Rombouts, Frederik
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 February 2013 23(3):785-790
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7 . Academic Journal
IMAGING ALZHEIMER'S TAU PATHOLOGY IN HUMANS: [18F]JNJ-067—A PHASE 0 EXPLORATORY STUDY IN HEALTHY VOLUNTEERS AND SUBJECTS WITH PROBABLE ALZHEIMER'S DISEASE
저자
by
Kolb, Hartmuth C.
;
Moechars, Diederik
;
Rombouts, Frederik
;
Schmidt, Mark E.
;
Szardenings, Anna Katrin
, et al.
소스
In
Alzheimer's & Dementia: The Journal of the Alzheimer's Association
July 2018 14(7) Supplement:P838-P838
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7 . Academic Journal
Direct nose to brain delivery of small molecules: critical analysis of data from a standardized in vivo screening model in rats.
저자
by
Dhuyvetter, Deborah
;
Tekle, Fetene
;
Nazarov, Maxim
;
Vreeken, Rob J.
;
Borghys, Herman
, et al.
소스
Drug Delivery
. Dec2020, Vol. 27 Issue 1, p1597-1607. 11p.
Open Access (T&F)
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7 . Academic Journal
Rational design and synthesis of aminopiperazinones as β-secretase (BACE) inhibitors
저자
by
Tresadern, Gary
;
Delgado, Francisca
;
Delgado, Oscar
;
Gijsen, Harrie
;
Macdonald, Gregor J.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2011 21(24):7255-7260
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7 . Periodical
Small-molecule BACE1 inhibitors: a patent literature review (2011 to 2020)
저자
by
Rombouts, Frederik
;
Kusakabe, Ken-ichi
;
Hsiao, Chien-Chi
;
Gijsen, Harrie J. M.
.
소스
Expert Opinion on Therapeutic Patents; January 2021, Vol. 31 Issue: 1 p25-52, 28p
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6 . Academic Journal
Preclinical Evaluation of
18
F-JNJ64349311, a Novel PET Tracer for Tau Imaging.
저자
by
Declercq, Lieven
;
Rombouts, Frederik
;
Koole, Michel
;
Fierens, Katleen
;
Mariën, Jonas
, et al.
소스
Journal of Nuclear Medicine; Jun2017, Vol. 58 Issue 6, p975-981, 7p, 1 Color Photograph, 1 Diagram, 2 Graphs
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