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1 . Academic Journal
Activation of Liver AMPK with PF-06409577 Corrects NAFLD and Lowers Cholesterol in Rodent and Primate Preclinical Models
저자
by
Ryan M. Esquejo
;
Christopher T. Salatto
;
Jake Delmore
;
Bina Albuquerque
;
Allan Reyes
, et al.
소스
EBioMedicine, Vol 31, Iss , Pp 122-132 (2018)
Full Text (ScienceDirect)
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7 .
6-Chloro-5-[4-(1-Hydroxycyclobutyl)Phenyl]-1H-Indole-3-Carboxylic Acid is a Highly Selective Substrate for Glucuronidation by UGT1A1, Relative toβ-Estradiol
저자
by
Kimberly Lapham
;
Jian Lin
;
Jonathan J. Novak
;
Heather Eng
;
Theunis C. Goosen
, et al.
소스
Drug Metabolism and Disposition
. 46:1836-1846
Open Access (OpenAIRE)
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7 .
Acyl Glucuronide Metabolites of 6-Chloro-5-[4-(1-hydroxycyclobutyl)phenyl]-1H-indole-3-carboxylic Acid (PF-06409577) and Related Indole-3-carboxylic Acid Derivatives are Direct Activators of Adenosine Monophosphate-Activated Protein Kinase (AMPK)
저자
by
Gregory S. Walker
;
Kimberly O. Cameron
;
Janice A. Brown
;
Daniel W. Kung
;
Angela Wolford
, et al.
소스
Journal of Medicinal Chemistry
. 61:7273-7288
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7 .
Activation of Liver AMPK with PF-06409577 Corrects NAFLD and Lowers Cholesterol in Rodent and Primate Preclinical Models
저자
by
Jessica Ward
;
Jason Barricklow
;
Chuong Nguyen
;
Eliza Bollinger
;
Christopher T. Salatto
, et al.
소스
EBioMedicine, Vol 31, Iss, Pp 122-132 (2018)
EBioMedicine
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7 .
Fall Armyworm: Impacts and Implications for Africa
저자
by
J. Godwin
;
Victor Attuquaye Clottey
;
Pablo González-Moreno
;
M. Bateman
;
Ivan Rwomushana
, et al.
소스
Outlooks on Pest Management
. 28:196-201
Scopus
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7 .
Selective Activation of AMPKβ1-Containing Isoforms Improves Kidney Function in a Rat Model of Diabetic Nephropathy
저자
by
Paul DaSilva-Jardine
;
Jessica Ward
;
Katherine Cialdea
;
Matthew F. Calabrese
;
Marina Amaro
, et al.
소스
Journal of Pharmacology and Experimental Therapeutics
. 361:303-311
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7 .
Recent progress in the identification of adenosine monophosphate-activated protein kinase (AMPK) activators
저자
by
Kimberly O. Cameron
;
Ravi G. Kurumbail
.
소스
Bioorganic & Medicinal Chemistry Letters
. 26:5139-5148
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4 .
Abstract 923: Pharmacological Activation of Ampk With a Direct Pan-ampk Activator Results in a Worsening of a Hf Phenotype in Mice
저자
by
Declan Flynn
;
Kimberly O. Cameron
;
Russell A. Miller
.
소스
Circulation Research
. 125
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5 .
Discovery and Preclinical Characterization of 6-Chloro-5-[4-(1-hydroxycyclobutyl)phenyl]-1H-indole-3-carboxylic Acid (PF-06409577), a Direct Activator of Adenosine Monophosphate-activated Protein Kinase (AMPK), for the Potential Treatment of Diabetic Nephropathy
저자
by
Jane M. Withka
;
Daniel W. Kung
;
Russell A. Miller
;
Matthew S. Dowling
;
Aaron C. Smith
, et al.
소스
Journal of Medicinal Chemistry
. 59:8068-8081
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7 .
Optimization of Metabolic and Renal Clearance in a Series of Indole Acid Direct Activators of 5'-Adenosine Monophosphate-Activated Protein Kinase (AMPK)
저자
by
Kimberly O. Cameron
;
Kevin J. Filipski
;
Jana Polivkova
;
Matthew S. Dowling
;
Andre Shavnya
, et al.
소스
Journal of medicinal chemistry
. 61(6)
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