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1 . Academic Journal
Discovery of Clinical Candidate GLPG3970: A Potent and Selective Dual SIK2/SIK3 Inhibitor for the Treatment of Autoimmune and Inflammatory Diseases.
저자
by
Peixoto, Christophe
;
Joncour, Agnes
;
Temal-Laib, Taouès
;
Tirera, Amynata
;
Dos Santos, Aurélie
, et al.
소스
Journal of Medicinal Chemistry; 4/11/2024, Vol. 67 Issue 7, p5233-5258, 26p
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7 . Periodical
Discovery, Structure–Activity Relationship, and Binding Mode of an Imidazo[1,2-a]pyridine Series of Autotaxin Inhibitors
저자
by
Joncour, Agnès
;
Desroy, Nicolas
;
Housseman, Christopher
;
Bock, Xavier
;
Bienvenu, Natacha
, et al.
소스
Journal of Medicinal Chemistry; 20240101, Issue: Preprints
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7 . Academic Journal
Discovery, Structure--Activity Relationship, and Binding Mode of an Imidazo[1,2-a]pyridine Series of Autotaxin Inhibitors.
저자
by
Joncour, Agnès
;
Desroy, Nicolas
;
Housseman, Christopher
;
Bock, Xavier
;
Bienvenu, Natacha
, et al.
소스
Journal of Medicinal Chemistry
. Sep2017, Vol. 60 Issue 17, p7371-7392. 22p.
Full Text (ACS)
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7 . Academic Journal
Discovery of 2-[[2-Ethyl-6-[4-[2-(3-hydroxyazetidin-1-yl)-2-oxoethyl]piperazin-1-yl]-8-methylimidazo[1,2-a]pyridin-3-yl]methylamino]-4-(4-fluorophenyl)thiazole-5-carbonitrile (GLPG1690), a First-in-Class Autotaxin Inhibitor Undergoing Clinical Evaluation for the Treatment of Idiopathic Pulmonary Fibrosis
저자
by
Desroy, Nicolas
;
Housseman, Christopher
;
Bock, Xavier
;
Joncour, Agnès
;
Bienvenu, Natacha
, et al.
소스
Journal of Medicinal Chemistry
. 5/11/2017, Vol. 60 Issue 9, p3580-3590. 11p.
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7 . Academic Journal
Synthesis of Anti-Microtubule Biaryls and Preliminary Evaluation as Vascular-Disrupting Agents.
저자
by
Joncour, Agnès
;
Liu, Jian-Miao
;
Décor, Anne
;
Thoret, Sylviane
;
Wdzieczak-Bakala, Joanna
, et al.
소스
ChemMedChem; 2008, Vol. 3 Issue 11, p1731-1739, 9p
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7 . Academic Journal
Asymmetric Synthesis of Antimicrotubule Biaryl Hybrids of Allocolchicine and Steganacin.
저자
by
Joncour, Agnès
;
Décor, Anne
;
Liu, Jian-Miao
;
Tran Huu Dau, Marie-Elise
;
Baudoin, Olivier
.
소스
Chemistry - A European Journal; Jun2007, Vol. 13 Issue 19, p5450-5465, 16p
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7 . Periodical
Biaryl Axis as a Stereochemical Relay for the Enantioselective Synthesis of Antimicrotubule Agents
저자
by
Joncour, Agnès
;
Décor, Anne
;
Thoret, Sylviane
;
Chiaroni, Angèle
;
Baudoin, Olivier
.
소스
Angewandte Chemie; June 2006, Vol. 118 Issue: 25 p4255-4258, 4p
Full Text (Wiley)
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7 . Academic Journal
Synthesis of antimicrotubule dibenzoxepines
저자
by
Colombel, Virginie
;
Joncour, Agnès
;
Thoret, Sylviane
;
Dubois, Joëlle
;
Bignon, Jérôme
, et al.
소스
Tetrahedron Letters: International Organ for the Rapid Publication of Preliminary Communications in Organic Chemistry
. Jun2010, Vol. 51 Issue 23, p3127-3129. 3p.
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7 . Academic Journal
Discovery, Structure Activity Relationship, and Binding Mode of an Imidazo[1,2-a]pyridine Series of Autotaxin Inhibitors (vol 60, pg 7371, 2017)
저자
by
Joncour, Agnes
;
Desroy, Nicolas
;
Housseman, Christopher
;
Bock, Xavier
;
Bienvenu, Natacha
, et al.
소스
JOURNAL OF MEDICINAL CHEMISTRY
; MAY 10 2018, 61 9, p4270-p4270, 1p.
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7 . Academic Journal
Discovery of GLPG1690: A first-in-class autotaxin inhibitor in clinical development for the treatment of idiopathic pulmonary fibrosis
저자
by
Desroy, Nicolas
;
Joncour, Agnes
;
Bock, Xavier
;
Housseman, Christopher
;
Peixoto, Christophe
, et al.
소스
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY
; MAR 13 2016, 251 1p.
Web of Science
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