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1 . Academic Journal
Discovery of a novel 2-spiroproline steroid mimetic scaffold for the potent inhibition of 11β-HSD1
저자
by
Burns, David M.
;
He, Chunhong
;
Li, Yun-Long
;
Zhuo, Jincong
;
Qian, Ding-Quan
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 October 2022 73
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7 . Academic Journal
Discovery of 1′-(1-phenylcyclopropane-carbonyl)-3H-spiro[isobenzofuran-1,3′-pyrrolidin]-3-one as a novel steroid mimetic scaffold for the potent and tissue-specific inhibition of 11β-HSD1 using a scaffold-hopping approach
저자
by
Zhang, Colin
;
Xu, Meizhong
;
He, Chunhong
;
Zhuo, Jincong
;
Burns, David M.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 August 2022 69
Full Text (ScienceDirect)
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7 . Academic Journal
High-Throughput Determination of Mode of Inhibition in Lead Identification and Optimization
저자
by
Wei, Min
;
Wynn, Richard
;
Hollis, Gregory
;
Liao, Boshan
;
Margulis, Alexander
, et al.
소스
In
SLAS Discovery
March 2007 12(2):220-228
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7 . Periodical
Discovery of Pemigatinib: A Potent and Selective Fibroblast Growth Factor Receptor (FGFR) Inhibitor
저자
by
Wu, Liangxing
;
Zhang, Colin
;
He, Chunhong
;
Qian, Dingquan
;
Lu, Liang
, et al.
소스
Journal of Medicinal Chemistry; August 2021, Vol. 64 Issue: 15 p10666-10679, 14p
Full Text (ACS)
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7 . Academic Journal
LSD1 Inhibition Induces Fetal Hemoglobin Expression and Provides a Novel Therapeutic Approach to Sickle Cell Disease
저자
by
Lee, Sang Hyun
;
Soloviev, Maxim
;
Zhang, Yan
;
Roman, Valerie
;
Yang, Gengjie
, et al.
소스
In
Blood
2 December 2016 128(22):2472-2472
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7 . Academic Journal
Conversion of an MMP-potent scaffold to an MMP-selective HER-2 sheddase inhibitor via scaffold hybridization and subtle [formula omitted] permutations
저자
by
Burns, David M.
;
He, Chunhong
;
Li, Yanlong
;
Scherle, Peggy
;
Liu, Xiangdong
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2008 18(2):560-564
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7 . Academic Journal
Design and identification of selective HER-2 sheddase inhibitors via P1′ manipulation and unconventional P2′ perturbations to induce a molecular metamorphosis
저자
by
Yao, Wenqing
;
Zhuo, Jincong
;
Burns, David M.
;
Li, Yun-Long
;
Qian, Ding-Quan
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2008 18(1):159-163
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7 . Academic Journal
A human CD137×PD-L1 bispecific antibody promotes anti-tumor immunity via context-dependent T cell costimulation and checkpoint blockade
저자
by
Geuijen, Cecile
;
Tacken, Paul
;
Wang, Liang-Chuan
;
Klooster, Rinse
;
van Loo, Pieter Fokko
, et al.
소스
Nature Communications
. 12(1)
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7 . Academic Journal
INCB054828 (pemigatinib), a potent and selective inhibitor of fibroblast growth factor receptors 1, 2, and 3, displays activity against genetically defined tumor models
저자
by
Liu, Phillip C. C.
;
Koblish, Holly
;
Wu, Liangxing
;
Bowman, Kevin
;
Diamond, Sharon
, et al.
소스
PLOS ONE
; APR 21 2020, 15 4, pe0231877 16p.
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7 . Academic Journal
Characterization of JAK2 V617F Allele Burden in Advanced Myelofibrosis (MF) Patients: No Change in V617F:WT JAK2 Ratio in Patients with High Allele Burdens despite Profound Clinical Improvement Following Treatment with the JAK Inhibitor, INCB018424
저자
by
Verstovsek, Srdan
;
Kantarjian, Hagop M.
;
Pardanani, Animesh D.
;
Burn, Timothy
;
Vaddi, Kris
, et al.
소스
In
Blood
16 November 2008 112(11):2802-2802
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