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1 . Academic Journal
AT7519, a Potent CDK Inhibitor, Is Active in Leukemia Models and Primary CLL Patient Samples.
저자
by
Squires, Matthew S.
;
Feltell, Ruth E.
;
Lock, Victoria
;
Smith, Donna M.
;
Lewis, Jon E.
, et al.
소스
In
Blood
16 November 2007 110(11):3127-3127
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7 . Academic Journal
AT13148 Is a Novel, Oral Multi-AGC Kinase Inhibitor with Potent Pharmacodynamic and Antitumor Activity
저자
by
Yap, Timothy A.
;
Walton, Mike I.
;
Grimshaw, Kyla M.
;
te Poele, Robert H.
;
Eve, Paul D.
, et al.
소스
CLINICAL CANCER RESEARCH
; JUL 15 2012, 18 14, p3912-p3923, 12p.
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7 . Academic Journal
Biological characterization of AT7519, a small-molecule inhibitor of cyclin-dependent kinases, in human tumor cell lines
저자
by
Squires, Matthew S.
;
Feltell, Ruth E.
;
Wallis, Nicola G.
;
Lewis, E. Jonathan
;
Smith, Donna-Michelle
, et al.
소스
MOLECULAR CANCER THERAPEUTICS
; FEB 2009, 8 2, p324-p332, 9p.
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7 . Academic Journal
Identification of N-(4-piperidinyl)-4-(2,6-dichlorobenzoylamino)-1H-pyrazole-3-carboxamide (AT7519), a novel cyclin dependent kinase inhibitor using fragment-based X-ray crystallography and structure based drug design
저자
by
Wyatt, Paul G.
;
Woodhead, Andrew J.
;
Berdini, Valerio
;
Boulstridge, John A.
;
Carr, Maria G.
, et al.
소스
JOURNAL OF MEDICINAL CHEMISTRY
; AUG 28 2008, 51 16, p4986-p4999, 14p.
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7 . Academic Journal
A comparison of the pharmacological profile of AT7519 in solid tumor and hematological cell lines
저자
by
Squires, Matthew S.
;
Feltell, Ruth E.
;
Lock, Victoria
;
Smith, Donna M.
;
Lewis, Ion E.
, et al.
소스
MOLECULAR CANCER THERAPEUTICS
; DEC 2007, 6 12, p3415S-p3416S, 2p.
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7 . Academic Journal
AT13148, an orally bioavailable AKT kinase inhibitor with potent anti-tumor activity in both in vitro and in vivo models exhibiting AKT pathway deregulation
저자
by
Lyons, John F.
;
Grimshaw, Kyla M.
;
Woodhead, Steven J.
;
Feltell, Ruth E.
;
Reule, Matthias
, et al.
소스
MOLECULAR CANCER THERAPEUTICS
; DEC 2007, 6 12, p3512S-p3512S, 1p.
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7 . Academic Journal
From fragment to lead: High throughput crystallography and rational design to identify CDKs inhibitors as anticancer drugs
저자
by
Berdini, Valerio
;
Boulstridge, John A.
;
Carr, Maria G.
;
Cross, David M.
;
Davis, Deborah J.
, et al.
소스
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY
; SEP 10 2006, 232 p142-p142, 1p.
Web of Science
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