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1 .
Discovery of a spirocyclic 3-bromo-4,5-dihydroisoxazole covalent inhibitor of hGAPDH with antiproliferative activity against pancreatic cancer cells
저자
by
Andrea Galbiati
;
Stefania Bova
;
Raffaella Pacchiana
;
Chiara Borsari
;
Marco Persico
, et al.
소스
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7 .
New Insights into the Structure–Activity Relationship and Neuroprotective Profile of Benzodiazepinone Derivatives of Neurounina-1 as Modulators of the Na+/Ca2+ Exchanger Isoforms
저자
by
Lucio Annunziato
;
Elisa Perissutti
;
Giuseppe Pignataro
;
Paolo Luciano
;
Agnese Secondo
, et al.
소스
Journal of Medicinal Chemistry
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7 .
Electronic Circular Dichroism Detects Conformational Changes Associated with Proteasome Gating Confirmed Using AFM Imaging
저자
by
Alessandro D’Urso
;
Roberto Purrello
;
Alessandra Cunsolo
;
Danilo Milardi
;
Caterina Fattorusso
, et al.
소스
Biomolecules; Volume 13; Issue 4; Pages: 704
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7 .
Modulation of the 20S Proteasome Activity by Porphyrin Derivatives Is Steered through Their Charge Distribution
저자
by
Marco Persico
;
Anna Maria Santoro
;
Alessandro D’Urso
;
Danilo Milardi
;
Roberto Purrello
, et al.
소스
Biomolecules; Volume 12; Issue 6; Pages: 741
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7 . Academic Journal
New antimalarial 3-methoxy-1,2-dioxanes: optimization of cellular pharmacokinetics and pharmacodynamics properties by incorporation of amino and N-heterocyclic moieties at C4.
저자
by
Sonawane, D. P.
;
Persico, M.
;
Corbett, Y.
;
Chianese, G.
;
Di Dato, A.
, et al.
소스
RSC Advances; 2015, Vol. 5 Issue 89, p72995-73010, 16p
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7 . Academic Journal
Marine inspired antiplasmodial thiazinoquinones: synthesis, computational studies and electrochemical assays.
저자
by
Imperatore, C.
;
Persico, M.
;
Aiello, A.
;
Luciano, P.
;
Guiso, M.
, et al.
소스
RSC Advances; 2015, Vol. 5 Issue 86, p70689-70702, 14p
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7 .
Tetra-substituted pyrrole derivatives act as potent activators of p53 in melanoma cells
저자
by
Paola Cuozzo
;
Giovanni Forte
;
Maria Pascale
;
Donatella Fiore
;
Maria Proto
, et al.
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Investigational New Drugs
. 38:634-649
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7 .
Hybrids between H2S-donors and betamethasone 17-valerate or triamcinolone acetonide inhibit mast cell degranulation and promote hyperpolarization of bronchial smooth muscle cells
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by
Ferdinando Fiorino
;
Marco Persico
;
Rocco Carmelo Pavese
;
Era Gorica
;
Francesco Petti
, et al.
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7 . Academic Journal
Outstanding effects on antithrombin activity of modified TBA diastereomers containing an optically pure acyclic nucleotide analogue.
저자
by
Scuotto, M.
;
Persico, M.
;
Bucci, M.
;
Vellecco, V.
;
Borbone, N.
, et al.
소스
Organic & Biomolecular Chemistry; 2014, Vol. 12 Issue 28, p5235-5242, 8p
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7 .
Cooperative Binding of the Cationic Porphyrin Tris-T4 Enhances Catalytic Activity of 20S Proteasome Unveiling a Complex Distribution of Functional States
저자
by
Roberto Purrello
;
Massimo Coletta
;
Marco Persico
;
Roberto Fattorusso
;
Diego Sbardella
, et al.
소스
International Journal of Molecular Sciences
Volume 21
Issue 19
International Journal of Molecular Sciences, Vol 21, Iss 7190, p 7190 (2020)
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