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1 . Academic Journal
Identification of Terfenadine as an Inhibitor of Human CD81-Receptor HCV-E2 Interaction: Synthesis and Structure Optimization
저자
by
Rolf W. Hartmann
;
Christian D. Klein
;
Lars Kattner
;
Ralf Bartenschlager
;
Artur Kaul
, et al.
소스
Molecules, Vol 13, Iss 5, Pp 1081-1110 (2008)
Open Access (DOAJ)
Web of Science
Scopus
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7 .
Corona versus Dengue: Distinct Mechanisms for Inhibition of Polyprotein Processing by Antiviral Drugs
저자
by
Mira A. M. Behnam
;
Christian D. Klein
.
소스
ACS Pharmacol Transl Sci
Open Access (OpenAIRE)
Scopus
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4 .
Discovery of potent benzoxaborole inhibitors against SARS-CoV-2 main and dengue virus proteases
저자
by
Nikos Kühl
;
Johannes Lang
;
Mila M. Leuthold
;
Christian D. Klein
.
소스
European journal of medicinal chemistry
. 240
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6 .
A New Class of Dengue and West Nile Virus Protease Inhibitors with Submicromolar Activity in Reporter Gene DENV-2 Protease and Viral Replication Assays
저자
by
Christian D. Klein
;
Nikos Kühl
;
Dominik Graf
;
Mila-Mareen Leuthold
;
Josephine Bock
, et al.
소스
Journal of Medicinal Chemistry
. 63:8179-8197
Web of Science
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7 .
Machine Learning in Mass Spectrometry: A MALDI-TOF MS Approach to Phenotypic Antibacterial Screening
저자
by
Luuk N. van Oosten
;
Christian D. Klein
.
소스
Journal of Medicinal Chemistry
. 63:8849-8856
Web of Science
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4 .
Diversity-oriented synthesis of peptide-boronic acids by a versatile building-block approach
저자
by
Christian D. Klein
;
Severin Kämmerer
;
Stefan P. A. Hinkes
.
소스
Chemical Science
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5 .
Inhibitor potency and assay conditions: A case study on SARS-CoV-2 main protease
저자
by
Christian D. Klein
;
Mira A. M. Behnam
.
소스
Proceedings of the National Academy of Sciences of the United States of America
Full Text (PNAS)
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Scopus
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4 .
The spectrum between substrates and inhibitors: Pinpointing the binding mode of dengue protease ligands with modulated basicity and hydrophobicity
저자
by
Christian D. Klein
;
Tonko Dražić
;
Nikos Kühl
;
Christina N Hacker
;
Nicole Gottscheber
.
소스
Bioorganicmedicinal chemistry
. 48
Scopus
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7 .
Insights into the design of inhibitors of the EGFR family with anticancer activity overcoming resistance: A case of optimizing thieno[2,3-d]pyrimidine-based EGFR inhibitors
저자
by
Sandra N. Milik
;
Amal Kamal Abdel-Aziz
;
Morad M. El-Hendawy
;
Riham I. El-Gogary
;
Mona Kamal Saadeldin
, et al.
소스
Journal of Molecular Structure
. 1259:132724
Web of Science
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7 . Academic Journal
Phenylalanine andPhenylglycine Analogues as ArginineMimetics in Dengue Protease Inhibitors.
저자
by
Lena F. Weigel
;
Christoph Nitsche
;
Dominik Graf
;
Ralf Bartenschlager
;
Christian D. Klein
.
소스
Journal of Medicinal Chemistry
. Oct2015, Vol. 58 Issue 19, p7719-7733. 15p.
Full Text (ACS)
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